TY - BOOK AU - AU - ED - SpringerLink (Online service) TI - Fragment-Based Drug Discovery and X-Ray Crystallography T2 - Topics in Current Chemistry, SN - 9783642275401 AV - QD415-436 U1 - 547 23 PY - 2012/// CY - Berlin, Heidelberg PB - Springer Berlin Heidelberg KW - Chemistry KW - Pharmaceutical technology KW - Chemistry, Organic KW - Crystallography KW - Organic Chemistry KW - Pharmaceutical Sciences/Technology N1 - D. A. Erlanson Introduction to Fragment-Based Drug Discovery -- T. G. Davies Ian J. Tickle Fragment Screening Using X-Ray Crystallography -- S. Roughley L. Wright P. Brough A. Massey R. E. Hubbard Hsp90 Inhibitors and Drugs from Fragment and Virtual Screening -- D. F. Wyss Y.-S. Wang H. L. Eaton C. Strickland J.s H. Voigt Z. Zhu A. W. Stamford Combining NMR and X-ray Crystallography in Fragment-Based Drug Discovery: Discovery of Highly Potent and Selective BACE-1 Inhibitors -- M. Hennig A. Ruf Walter HuberCombining Biophysical Screening and X-Ray Crystallography for Fragment-Based Drug Discovery -- E. Valkov T. Sharpe M. Marsh Sa. Greive M. Hyvȵnen Targeting ProteinProtein Interactions and Fragment-Based Drug Discovery -- J.h D. Bauman D. Patel E. Arnold Fragment Screening and HIV Therapeutics -- D. Rognan Fragment-Based Approaches and Computer-Aided Drug Discovery; ZDB-2-CMS N2 - D. A. Erlanson Introduction to Fragment-Based Drug Discovery T. G. Davies Ian J. Tickle Fragment Screening Using X-Ray Crystallography S. Roughley L. Wright P. Brough A. Massey R. E. Hubbard Hsp90 Inhibitors and Drugs from Fragment and Virtual Screening D. F. Wyss Y.-S. Wang H. L. Eaton C. Strickland J.s H. Voigt Z. Zhu A. W. Stamford Combining NMR and X-ray Crystallography in Fragment-Based Drug Discovery: Discovery of Highly Potent and Selective BACE-1 Inhibitors M. Hennig A. Ruf Walter HuberCombining Biophysical Screening and X-Ray Crystallography for Fragment-Based Drug Discovery E. Valkov T. Sharpe M. Marsh Sa. Greive M. Hyvȵnen Targeting ProteinProtein Interactions and Fragment-Based Drug Discovery J.h D. Bauman D. Patel E. Arnold Fragment Screening and HIV Therapeutics D. Rognan Fragment-Based Approaches and Computer-Aided Drug Discovery UR - http://dx.doi.org/10.1007/978-3-642-27540-1 ER -